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Tesmilifene fumarate
CAS No. 1185241-83-1
Tesmilifene fumarate ( DPPE fumarate )
产品货号. M23352 CAS No. 1185241-83-1
Tesmifene fumarate (DPPE fumarate) 是一种 H1C 受体拮抗剂。
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| 规格 | 价格/人民币 | 库存 | 数量 |
| 2MG | ￥223 | 有现货 |
|
| 5MG | ￥373 | 有现货 |
|
| 10MG | ￥568 | 有现货 |
|
| 25MG | ￥995 | 有现货 |
|
| 50MG | ￥1609 | 有现货 |
|
| 100MG | ￥2304 | 有现货 |
|
| 200MG | ￥3285 | 有现货 |
|
| 500MG | 获取报价 | 有现货 |
|
| 1G | 获取报价 | 有现货 |
|
| 1 mL x 10 mM in DMSO | ￥426 | 有现货 |
|
生物学信息
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产品名称Tesmilifene fumarate
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注意事项本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
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产品简述Tesmifene fumarate (DPPE fumarate) 是一种 H1C 受体拮抗剂。
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产品描述Tesmilifene fumarate (DPPE fumarate) is an H1C receptor antagonist。
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体外实验Tesmilifene may modulate the effects of 12(S)HETE in cancer cells, and indirectly, influence the susceptibility of cellular DNA to chemotherapy.
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体内实验Tesmilifene (DPPE, 20 mg/kg (s.c.) and 20 μg (icv in 5 μL)) potentiated seizures induced by both convulsants. Animal Model:Male BKTO mice (25-45 g).Dosage:20 mg/kg (s.c.) and 20 μg (icv in 5 μL).Administration:S.C. and icv.Result:Potentiated seizures induced by both convulsants.
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同义词DPPE fumarate
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通路GPCR/G Protein
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靶点Histamine Receptor
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受体Histamine Receptor
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研究领域——
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适应症——
化学信息
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CAS Number1185241-83-1
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分子量399.48
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分子式C23H29NO5
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纯度>98% (HPLC)
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溶解度DMSO:248 mg/mL (620.81 mM; Need ultrasonic)
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SMILESCCN(CC)CCOC1=CC=C(C=C1)CC2=CC=CC=C2.OC(/C=C/C(O)=O)=O
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化学全称——
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1.Mark Vincent, et al. Tesmilifene may enhance breast cancer chemotherapy by killing a clone of aggressive, multi-drug resistant cells through its action on the p-glycoprotein pump. Med Hypotheses. 2006;66(4):715-31.
产品手册
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