Activator of protein kinase C; attached to cell permeabilization Antennapedia domain vector peptide. Consists of peptide derived from the C2 domain of PKC β linked by a disulfide bridge to the Antennapedia domain vector peptide. The Antennapedia peptide is actively taken up by intact cells, at 4 or 37°C, ensuring rapid and effective uptake of the activator peptide. Once inside the cell, the disulfide bonds are subjected to reduction in the cytoplasm leading to release of the activator peptide.

苯胺芥子是具有抗肿瘤活性的烷基化芥子。

4-噻唑甲酰胺，N-[2-[(2S)-2-氰基-4,4-二氟-1-吡咯烷基]-2-氧代乙基]-2-[(3,4-二氯苯基)甲基]-(BR102910)是成纤维细胞激活蛋白（FAP）的选择性抑制剂。