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Dalcotidine
CAS No. 120958-90-9
Dalcotidine ( —— )
产品货号. M34564 CAS No. 120958-90-9
Dalcotidine (KU 1257) is a novel histamine H2 receptor antagonist with histamine H9 receptor antagonistic activity and antisecretory effects.The Ki value for binding to guinea pig cerebral cortex was 0.040 The KB value for antagonism of histamine-induced positive chronotropic responses in the right atrium of isolate guinea pigs was 0.041.Dalcotidine improves the quality of ulcer healing, and may contribute to a reduction in ulcer recurrence and relapse rates.
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| 规格 | 价格/人民币 | 库存 | 数量 |
| 5MG | ￥979 | 有现货 |
|
| 10MG | ￥1482 | 有现货 |
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| 25MG | ￥2334 | 有现货 |
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| 50MG | ￥3367 | 有现货 |
|
| 100MG | ￥4617 | 有现货 |
|
| 200MG | ￥6219 | 有现货 |
|
| 500MG | 获取报价 | 有现货 |
|
| 1G | 获取报价 | 有现货 |
|
| 1 mL x 10 mM in DMSO | ￥938 | 有现货 |
|
生物学信息
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产品名称Dalcotidine
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注意事项本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
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产品简述Dalcotidine (KU 1257) is a novel histamine H2 receptor antagonist with histamine H9 receptor antagonistic activity and antisecretory effects.The Ki value for binding to guinea pig cerebral cortex was 0.040 The KB value for antagonism of histamine-induced positive chronotropic responses in the right atrium of isolate guinea pigs was 0.041.Dalcotidine improves the quality of ulcer healing, and may contribute to a reduction in ulcer recurrence and relapse rates.
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产品描述Dalcotidine (KU 1257) is a novel histamine H2 receptor antagonist with histamine H9 receptor antagonistic activity and antisecretory effects.The Ki value for binding to guinea pig cerebral cortex was 0.040 The KB value for antagonism of histamine-induced positive chronotropic responses in the right atrium of isolate guinea pigs was 0.041.Dalcotidine improves the quality of ulcer healing, and may contribute to a reduction in ulcer recurrence and relapse rates.
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体外实验——
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体内实验——
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同义词——
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通路GPCR/G Protein
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靶点Histamine Receptor
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受体Histamine Receptor
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研究领域——
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适应症——
化学信息
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CAS Number120958-90-9
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分子量319.44
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分子式C18H29N3O2
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纯度>98% (HPLC)
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溶解度——
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SMILESC(C1=CC(OCCCNC(NCC)=O)=CC=C1)N2CCCCC2
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化学全称——
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
产品手册
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