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Ticolubant
CAS No. 154413-61-3
Ticolubant ( —— )
产品货号. M34447 CAS No. 154413-61-3
Ticolubant is orally active leukotriene B4 antagonist with high affinity for the human neutrophil LTB4 receptor (Ki = 0.78 nM), blocks LTB4-induced Ca2+ migration with an IC50 of 6.6 ± 1.5 nM, and shows topical anti-inflammatory activity in a mouse model of skin inflammation.
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| 规格 | 价格/人民币 | 库存 | 数量 |
| 5MG | ￥2100 | 有现货 |
|
| 10MG | ￥3012 | 有现货 |
|
| 25MG | ￥4585 | 有现货 |
|
| 50MG | ￥6398 | 有现货 |
|
| 100MG | ￥8523 | 有现货 |
|
| 200MG | ￥11430 | 有现货 |
|
| 500MG | 获取报价 | 有现货 |
|
| 1G | 获取报价 | 有现货 |
|
生物学信息
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产品名称Ticolubant
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注意事项本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
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产品简述Ticolubant is orally active leukotriene B4 antagonist with high affinity for the human neutrophil LTB4 receptor (Ki = 0.78 nM), blocks LTB4-induced Ca2+ migration with an IC50 of 6.6 ± 1.5 nM, and shows topical anti-inflammatory activity in a mouse model of skin inflammation.
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产品描述Ticolubant is orally active leukotriene B4 antagonist with high affinity for the human neutrophil LTB4 receptor (Ki = 0.78 nM), blocks LTB4-induced Ca2+ migration with an IC50 of 6.6 ± 1.5 nM, and shows topical anti-inflammatory activity in a mouse model of skin inflammation.
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体外实验——
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体内实验——
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同义词——
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通路GPCR/G Protein
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靶点Calcium Channel
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受体Calcium Channel | LTR
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研究领域——
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适应症——
化学信息
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CAS Number154413-61-3
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分子量460.37
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分子式C23H19Cl2NO3S
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纯度>98% (HPLC)
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溶解度——
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SMILESC(=C/C(O)=O)\C1=C(OCCC2=CC=CC=C2)C=CC(CSC3=C(Cl)C=CC=C3Cl)=N1
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化学全称——
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
产品手册
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