Ninerafaxstat 使细胞代谢从脂肪酸氧化转向葡萄糖氧化。Ninerafaxstat 减少脂肪酸氧化并改善整体线粒体呼吸。Ninerafaxstat 抑制癌细胞的生长和增殖。

Silybin B is an effective inhibitor of raloxifene 4 '- and 6-glucosalylation, an effective anti-fibrinogenic and anti-oligomeric component of Silymarin, with free radical scavenging activity of 1, 1-diphenyl-2-pyridinyl hydrazine (DPPH), and a protective effect against cisplatin-induced neurotoxicity by alleviating DNA damage and apoptosis.

GAK抑制剂49是一种高度选择性和ATP竞争性的细胞周期蛋白G相关激酶（GAK）抑制剂（IC50：56 nM；Ki：0.54 nM）。