Obtusin ( —— )

产品货号. M29200 CAS No. 70588-05-5

COA

Datasheet

HNMR

HPLC

MSDS

Handing Instructions

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产品名称

Obtusin
注意事项

本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
产品简述

Obtusin 是来自决明子种子，是一种高度选择性和竞争性的人单胺氧化酶-A (hMAO-A) 抑制剂，IC50 为 11.12 μM，Ki 为 6.15 μM。Obtusin 在神经退行性疾病，尤其是焦虑和抑郁中起预防作用。
产品描述

Obtusin is a natural product.(In Vitro):Nine anthraquinones, aurantio-Obtusin (1), chryso-Obtusin (2), Obtusin (3), chryso-Obtusin-2-O-beta-D-glucoside (4), physcion (5), emodin (6), chrysophanol (7), obtusifolin (8), and obtusifolin-2-O-beta-D-glucoside (9), isolated from an EtOAc-soluble extract of the seeds of Cassia tora, were subjected to in vitro bioassays to evaluate their inhibitory activity against advanced glycation end products (AGEs) formation and rat lens aldose reductase (RLAR).
体外实验

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体内实验

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同义词

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通路

Metabolic Enzyme/Protease
靶点

MAO
受体

MAO
研究领域

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适应症

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计算器

产品手册

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