021-51111890
购物车（）
sales@molnova.cn
Metiamide
CAS No. 34839-70-8
Metiamide ( SK&F 92058 )
产品货号. M20781 CAS No. 34839-70-8
Metiamide 是一种组胺 H2 受体拮抗剂。
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| 规格 | 价格/人民币 | 库存 | 数量 |
| 5MG | ￥1416 | 有现货 |
|
| 10MG | ￥2261 | 有现货 |
|
| 25MG | ￥3469 | 有现货 |
|
| 50MG | ￥4604 | 有现货 |
|
| 100MG | ￥7092 | 有现货 |
|
| 500MG | 获取报价 | 有现货 |
|
| 1G | 获取报价 | 有现货 |
|
| 1 mL x 10 mM in DMSO | ￥1264 | 有现货 |
|
生物学信息
-
产品名称Metiamide
-
注意事项本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
-
产品简述Metiamide 是一种组胺 H2 受体拮抗剂。
-
产品描述Metiamide is a histamine H2-receptor antagonist .
-
体外实验Metiamide (SK&F 92058) is a competitivewith aldehyde substrates and noncompetitive with the Human E3 Aldehyde Dehydrogenase coenzyme, binding to both the free E3 isozyme and the enzyme·coenzyme binary complex with Ki values of 0.92 μM glycolaldehyde as the varied substrate. Data is got as percentage change in GTPase activity induced by metiamide compared with the GTPase activity stimulated by HA (100 μM).
-
体内实验——
-
同义词SK&F 92058
-
通路GPCR/G Protein
-
靶点Histamine Receptor
-
受体H2 receptor
-
研究领域——
-
适应症——
化学信息
-
CAS Number34839-70-8
-
分子量244.38
-
分子式C9H16N4S2
-
纯度>98% (HPLC)
-
溶解度DMSO:2.4 mg/mL (9.82 mM)
-
SMILESCNC(=S)NCCSCc1[nH]cnc1C
-
化学全称1-methyl-3-(2-(((5-methyl-1H-imidazol-4-yl)methyl)thio)ethyl)thiourea
运输与储存
-
储存条件(-20℃)
-
运输条件With Ice Pack
-
稳定性≥ 2 years
参考文献
1.Blair E L Grund E R Miller I T et al. Metiamide in the Zollinger-Ellison syndrome[J]. The American Journal of Digestive Diseases 1976 20(12):1123-1130.
产品手册
关联产品
-
Antazoline hydrochlo...
盐酸安他唑啉是第一代抗组胺药，与组胺 H1 受体结合并阻断内源性组胺的作用。
-
Efletirizine
Efletirizine (UCB-28754) is a histamine receptor antagonist with inhibitory effects on the enzyme 5-lipoxygenase (5-LO), and is useful in the topical treatment of allergic diseases.
-
Tecastemizole
Tecastimizole 是 H1 受体的选择性拮抗剂，是阿司咪唑的主要代谢产物，具有抗炎作用。
