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GSK1940029

CAS No. 1150701-66-8

GSK1940029 ( SCD inhibitor 1 )

产品货号. M20222 CAS No. 1150701-66-8

GSK1940029 是一种硬脂酰辅酶去饱和酶 (SCD) 抑制剂。

纯度: >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
规格 价格/人民币 库存 数量
5MG ¥1492 有现货
10MG ¥2176 有现货
25MG ¥3692 有现货
50MG ¥5450 有现货
100MG ¥7092 有现货
200MG ¥9540 有现货
500MG 获取报价 有现货
1G 获取报价 有现货
1 mL x 10 mM in DMSO ¥1511 有现货

生物学信息

  • 产品名称
    GSK1940029
  • 注意事项
    本公司产品仅用于科研实验,不得用于人体或动物的临床与诊断
  • 产品简述
    GSK1940029 是一种硬脂酰辅酶去饱和酶 (SCD) 抑制剂。
  • 产品描述
    GSK1940029 is a stearoyl-coa desaturase (SCD) inhibitor.(In Vitro):GSK1940029 (SCD inhibitor 1) is a stearoyl-coa desaturase (SCD), which can be used to treat and/or preventing various diseases, including those mediated by SCD enzyme, such as diseases related to elevated lipid levels, cardiovascular disease, diabetes, obesity, metabolic syndrome, skin disorders such as acne, diseases or conditions related to cancer and the treatment of symptoms linked to the production of the amyloid plaque-forming Aβ42 peptide such as Alzheimer's disease.
  • 体外实验
    GSK1940029 (SCD inhibitor 1) is a stearoyl-coa desaturase (SCD), which can be used to treat and/or preventing various diseases, including those mediated by SCD enzyme, such as diseases related to elevated lipid levels, cardiovascular disease, diabetes, obesity, metabolic syndrome, skin disorders such as acne, diseases or conditions related to cancer and the treatment of symptoms linked to the production of the amyloid plaque-forming Aβ42 peptide such as Alzheimer's disease.
  • 体内实验
    ——
  • 同义词
    SCD inhibitor 1
  • 通路
    Metabolic Enzyme/Protease
  • 靶点
    Dehydrogenase
  • 受体
    SCD
  • 研究领域
    Endocrinology
  • 适应症
    Acne Vulgaris

化学信息

  • CAS Number
    1150701-66-8
  • 分子量
    391.25
  • 分子式
    C18H16Cl2N4O2
  • 纯度
    >98% (HPLC)
  • 溶解度
    DMSO:30 mg/mL (76.67 mM)
  • SMILES
    Cc1c(nnn1Cc1ccc(Cl)c(Cl)c1)C(=O)Nc1ccc(CO)cc1
  • 化学全称
    1-[(34-dichlorophenyl)methyl]-N-[4-(hydroxymethyl)phenyl]-5-methyltriazole-4-carboxamide

运输与储存

  • 储存条件
    (-20℃)
  • 运输条件
    With Ice Pack
  • 稳定性
    ≥ 2 years

参考文献

1.Anne Marie Jeanne Bouillot et al. 1 2 3-triazole derivatives for use as stearoyl-coa desaturase inhibitors . PCT Int. Appl. (2009) WO 2009060053 A1 20090514.
产品手册
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