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Nafronyl oxalate

CAS No. 3200-06-4

Nafronyl oxalate ( Nafronyl Oxalate | Dubimax: Dusodril: Naftidrofuryl oxalate )

产品货号. M14041 CAS No. 3200-06-4

一种用于治疗外周和脑血管疾病的化合物。据称它可以增强细胞氧化能力并具有解痉作用。

纯度: >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
规格 价格/人民币 库存 数量
50MG ¥219 有现货
100MG ¥372 有现货
200MG ¥529 有现货
500MG ¥882 有现货
1G 获取报价 有现货
1 mL x 10 mM in DMSO ¥145 有现货

生物学信息

  • 产品名称
    Nafronyl oxalate
  • 注意事项
    本公司产品仅用于科研实验,不得用于人体或动物的临床与诊断
  • 产品简述
    一种用于治疗外周和脑血管疾病的化合物。据称它可以增强细胞氧化能力并具有解痉作用。
  • 产品描述
    A drug used in the management of peripheral and cerebral vascular disorders. It is claimed to enhance cellular oxidative capacity and to be a spasmolytic. (From Martindale, The Extra Pharmacopoeia, 30th ed, p1310) It may also be an antagonist at 5HT-2 serotonin receptors. (In Vitro):Naftidrofuryl oxalate (Nafronyl oxalate salt) may be effective for relieving the pain of muscle cramps.Naftidrofuryl oxalate (Nafronyl oxalate salt) is the only vasoactive drug for peripheral arterial disease (PAD) which is likely to be cost-effective.Naftidrofuryl oxalate (Nafronyl oxalate salt) is ranked first for both maximum walking distance (MWD) and pain-free walking distance (PFWD) (probability of 0·947 and 0·987, respectively, of being the best treatment) followed by cilostazol and pentoxifylline. Naftidrofuryl oxalate (Nafronyl oxalate salt) is effective treatments for claudication, Naftidrofuryl oxalate is likely to be the most effective, with minimal serious adverse events.
  • 体外实验
    Naftidrofuryl oxalate (Nafronyl oxalate salt) may be effective for relieving the pain of muscle cramps.Naftidrofuryl oxalate (Nafronyl oxalate salt) is the only vasoactive drug for peripheral arterial disease (PAD) which is likely to be cost-effective.Naftidrofuryl oxalate (Nafronyl oxalate salt) is ranked first for both maximum walking distance (MWD) and pain-free walking distance (PFWD) (probability of 0·947 and 0·987, respectively, of being the best treatment) followed by cilostazol and pentoxifylline. Naftidrofuryl oxalate (Nafronyl oxalate salt) is effective treatments for claudication, Naftidrofuryl oxalate is likely to be the most effective, with minimal serious adverse events.
  • 体内实验
    ——
  • 同义词
    Nafronyl Oxalate | Dubimax: Dusodril: Naftidrofuryl oxalate
  • 通路
    Endocrinology/Hormones
  • 靶点
    5-HT Receptor
  • 受体
    5-HT
  • 研究领域
    Cardiovascular Disease
  • 适应症
    ——

化学信息

  • CAS Number
    3200-06-4
  • 分子量
    473.56
  • 分子式
    C26H35NO7
  • 纯度
    >98% (HPLC)
  • 溶解度
    Water: 10 mM
  • SMILES
    O=C(OCCN(CC)CC)C(CC1=C2C=CC=CC2=CC=C1)CC3OCCC3.O=C(O)C(O)=O
  • 化学全称
    2-(Diethylamino)ethyl 2-(naphthalen-1-ylmethyl)-3-(oxolan-2-yl)propanoate Oxalate

运输与储存

  • 储存条件
    (-20℃)
  • 运输条件
    With Ice Pack
  • 稳定性
    ≥ 2 years

参考文献

1. Kim MJ, et al. Clin Exp Nephrol. 2013 Jun;17(3):437-8.
产品手册
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