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CL 316243
CAS No. 183720-02-7
CL 316243 ( BTA 243 )
产品货号. M12836 CAS No. 183720-02-7
CL 316243 (BTA 243) 是一种有效的、高选择性的、口服活性的 β3-肾上腺素受体激动剂，EC50 为 3 nM。
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| 规格 | 价格/人民币 | 库存 | 数量 |
| 25MG | ￥15531 | 有现货 |
|
| 50MG | ￥20925 | 有现货 |
|
| 100MG | ￥25830 | 有现货 |
|
| 500MG | 获取报价 | 有现货 |
|
| 1G | 获取报价 | 有现货 |
|
生物学信息
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产品名称CL 316243
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注意事项本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
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产品简述CL 316243 (BTA 243) 是一种有效的、高选择性的、口服活性的 β3-肾上腺素受体激动剂，EC50 为 3 nM。
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产品描述CL 316243 (BTA 243) is a potent, highly selective, orally active β3-adrenoceptor agonist with EC50 of 3 nM; Displays >10000-fold selective over β1 and β2 receptors; Significantly increases brown adipose tissue thermogenesis and resting metabolic rate in mice, also increases the concentration of insulin receptors and decreases the levels of serum insulin and blood glucose during the glucose overloading test.Obesity Discontinued.
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体外实验——
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体内实验——
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同义词BTA 243
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通路GPCR/G Protein
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靶点Adrenergic Receptor
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受体Adrenergic Receptor
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研究领域Metabolic Disease
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适应症Obesity
化学信息
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CAS Number183720-02-7
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分子量421.83
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分子式C20H20ClNO7
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纯度>98% (HPLC)
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溶解度——
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SMILESCC(CC1=CC2=C(C=C1)OC(O2)(C(=O)O)C(=O)O)NCC(C3=CC(=CC=C3)Cl)O
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化学全称5-[(2R)-2-[[(2R)-2-(3-Chlorophenyl)-2-hydroxyethyl]amino]propyl]-1,3-benzodioxole-2,2-dicarboxylic acid
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1. Berlan M, et al. J Pharmacol Exp Ther. 1994 Mar;268(3):1444-51.
2. Himms-Hagen J, et al. Am J Physiol. 1994 Apr;266(4 Pt 2):R1371-82.
3. Yoshida T, et al. Life Sci. 1994;54(7):491-8.
产品手册
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