Highly potent integrin α1β1 inhibitor (IC50 = 0.8 nM for α1β1 binding to type IV collagen). Selective for α1β1 over α2β1, αIIbβ3, αvβ3, α4β1, α5β6, α9β1 and α4β7. Inhibits FGF2-stimulated angiogenesis in the chicken chorioallantoic model. Displays antitumor efficacy in a synergistic mouse model of Lewis lung carcinoma; blocks human melanoma growth in nude mice.

依托贝特是氯贝特和烟酸的组合，用于治疗高脂血症。

Chrysophanol 8-O-β-D-(6’-O-galloyl)glucopyranoside 是一种蒽醌葡萄糖苷，可以从 Rheum undulatum L 中分离出来。Chrysophanol 8-O-β-D-(6’-O-galloyl)glucopyranoside 具有有效的 DPPH 自由基和 O2- 清除活性。