
ROS kinases-IN-1
CAS No. 370096-57-4
ROS kinases-IN-1 ( —— )
产品货号. M35383 CAS No. 370096-57-4
ROS kinases-IN-1 (pag 98) 是一种 ROS 酪氨酸激酶抑制剂,IC50 值为 1.22 μM。ROS kinases-IN-1 具有抗肿瘤活性。
纯度: >98% (HPLC)






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生物学信息
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产品名称ROS kinases-IN-1
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注意事项本公司产品仅用于科研实验,不得用于人体或动物的临床与诊断
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产品简述ROS kinases-IN-1 (pag 98) 是一种 ROS 酪氨酸激酶抑制剂,IC50 值为 1.22 μM。ROS kinases-IN-1 具有抗肿瘤活性。
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产品描述ROS kinases-IN-1 (pag 98) is a ROS tyrosine kinase inhibitor with IC50 value of 1.22 μM. ROS kinases-IN-1 shows anti-tumor activity.
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体外实验ROS kinases-IN-1 (1-100 μM; 1 d) inhibits the growth of cervical cancer cell and glioblastoma cells.Cell Viability Assay Cell Line:HeLa, U138, U87, LN18, and U118 cells Concentration:1, 10, and 100 μM Incubation Time:one day Result:Showed EC50s for HeLa, U138, U87, LN18, and U118 cells of 20, 8, 8, 12, and 7 μM, respectively.
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体内实验——
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同义词——
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通路Immunology/Inflammation
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靶点ROS
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受体ROS Kinase
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研究领域——
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适应症——
化学信息
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CAS Number370096-57-4
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分子量328.37
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分子式C20H16N4O
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纯度>98% (HPLC)
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溶解度In Vitro:?DMSO 中的溶解度 : 20.83 mg/mL (63.43 mM; 超声助溶 (<60°C)
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SMILESCC1=NNC(=O)\C1=C\c1cn(nc1-c1ccccc1)-c1ccccc1
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化学全称——
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1. Dorre A. GRUENEBERG, et al. Novel methods, compounds, and compositions for inhibition of ros. WO2014141129A2.
产品手册




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