
Pirodomast
CAS No. 108310-20-9
Pirodomast ( —— )
产品货号. M36113 CAS No. 108310-20-9
Pirodomast is a thromboxane A (TXA2) synthase inhibitor. Pirodomast inhibits leukotriene (LT) D4, C4, E4 formation and thromboxane B2 (TXB2) activity, but is weakly or ineffectively antagonistic to guinea pig bronchospasm induced by histamine, methacholine, serotonin, LTC4, or platelet-activating factor.
纯度: >98% (HPLC)






规格 | 价格/人民币 | 库存 | 数量 |
2MG | ¥2093 | 有现货 |
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5MG | ¥3149 | 有现货 |
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10MG | ¥4764 | 有现货 |
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25MG | ¥7374 | 有现货 |
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50MG | ¥10010 | 有现货 |
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100MG | ¥13235 | 有现货 |
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500MG | ¥26469 | 有现货 |
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1G | 获取报价 | 有现货 |
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生物学信息
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产品名称Pirodomast
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注意事项本公司产品仅用于科研实验,不得用于人体或动物的临床与诊断
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产品简述Pirodomast is a thromboxane A (TXA2) synthase inhibitor. Pirodomast inhibits leukotriene (LT) D4, C4, E4 formation and thromboxane B2 (TXB2) activity, but is weakly or ineffectively antagonistic to guinea pig bronchospasm induced by histamine, methacholine, serotonin, LTC4, or platelet-activating factor.
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产品描述Pirodomast is a thromboxane A (TXA2) synthase inhibitor. Pirodomast inhibits leukotriene (LT) D4, C4, E4 formation and thromboxane B2 (TXB2) activity, but is weakly or ineffectively antagonistic to guinea pig bronchospasm induced by histamine, methacholine, serotonin, LTC4, or platelet-activating factor. Pirodomast is a potential antiallergic compound. Pirodomast had only weak relaxant activity on guinea pig trachea in vitro. Pirodomast is a potential antiallergic compound that inhibits the protein hydrolyzing activity of trypsin in vitro, prevents antigen-induced immediate and late asthmatic responses in allergic sheep in vivo, and inhibits antigen-induced airway hyperresponsiveness to histamine and carbachol in allergic sheep.
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体外实验——
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体内实验——
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同义词——
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通路Autophagy
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靶点Thrombin
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受体Thrombin | Serine Protease
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研究领域——
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适应症——
化学信息
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CAS Number108310-20-9
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分子量307.35
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分子式C18H17N3O2
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纯度>98% (HPLC)
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溶解度——
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SMILESO=C1N(C=2C(C(=O)C1N3CCCC3)=CC=CN2)C4=CC=CC=C4
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化学全称——
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
产品手册




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