Potent GPR37L1 and GPR37 agonist (EC50 values are 5 and 7 nM, respectively). Stimulates signaling through pertussis toxin-sensitive G proteins. Stimulates ERK phosphorylation. Protects against cellular stress. Promotes myelin lipid synthesis and prolongs cell survival in both Schwann cells and oligodendrocytes; neuroprotective and glioprotective.

SR11237 是一种泛视黄醇 X 受体 (RXR) 激动剂。 SR11237 导致 RXR/RXR 同二聚体形成并反式激活含有 RXR 响应元件的报告基因。

DL-α-(Difluoromethyl)arginine 是一种有效的酶激活且不可逆的精氨酸脱羧酶抑制剂。DL-α-(Difluoromethyl)arginine 可阻断体内 E.coli 和 Pseudomonas aeruginosa 的精氨酸脱羧酶活性。