Tat-NR2B9c (NA-1) 是一种神经保护剂；与 PSD-95 的第二个 PDZ 结构域表现出高亲和力结合。

Apelin biased agonist; exhibits bias for the G protein pathway. Stimulates endothelial NOS phosphorylation and expression, promotes proliferation, and attenuates apoptosis of human pulmonary arterial endothelial cells in vitro. Shows positive inotropic and vasodilatory effects in vivo and improves cardiac structure and function in a model of pulmonary arterial hypertension.

MD2-IN-1 是一种骨髓分化蛋白 2 (MD2) 抑制剂，对重组人 MD2 (rhMD2) 的 KD 为 189 μM。