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Dehydro Nifedipine
CAS No. 67035-22-7
Dehydro Nifedipine ( —— )
产品货号. M34871 CAS No. 67035-22-7
Dehydro Nifedipine (BAY-b 4759) is the main metabolite of nifedipine in human plasma. Dehydro Nifedipine inhibits glucose uptake in PC-12 cells with an IC50 value of 130 μM. Nifedipine is a calcium channel blocker used in the treatment of hypertension and angina. Dehydronifedipine is formed when it is metabolized by cytochrome P450 (CYP) isomers CYP3A4 and CYP3A5.
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| 规格 | 价格/人民币 | 库存 | 数量 |
| 5MG | ￥392 | 有现货 |
|
| 10MG | ￥629 | 有现货 |
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| 25MG | ￥1228 | 有现货 |
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| 50MG | ￥1944 | 有现货 |
|
| 100MG | ￥3024 | 有现货 |
|
| 200MG | ￥4302 | 有现货 |
|
| 500MG | 获取报价 | 有现货 |
|
| 1G | 获取报价 | 有现货 |
|
生物学信息
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产品名称Dehydro Nifedipine
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注意事项本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
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产品简述Dehydro Nifedipine (BAY-b 4759) is the main metabolite of nifedipine in human plasma. Dehydro Nifedipine inhibits glucose uptake in PC-12 cells with an IC50 value of 130 μM. Nifedipine is a calcium channel blocker used in the treatment of hypertension and angina. Dehydronifedipine is formed when it is metabolized by cytochrome P450 (CYP) isomers CYP3A4 and CYP3A5.
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产品描述Dehydro Nifedipine (BAY-b 4759) is the main metabolite of nifedipine in human plasma. Dehydro Nifedipine inhibits glucose uptake in PC-12 cells with an IC50 value of 130 μM. Nifedipine is a calcium channel blocker used in the treatment of hypertension and angina. Dehydronifedipine is formed when it is metabolized by cytochrome P450 (CYP) isomers CYP3A4 and CYP3A5.
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体外实验——
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体内实验——
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同义词——
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通路Others
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靶点Other Targets
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受体Drug Metabolite
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研究领域——
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适应症——
化学信息
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CAS Number67035-22-7
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分子量344.32
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分子式C17H16N2O6
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纯度>98% (HPLC)
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溶解度——
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SMILESCOC(=O)c1c(C)nc(C)c(C(=O)OC)c1-c1ccccc1[N+]([O-])=O
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化学全称——
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
产品手册
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