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Rilmakalim
CAS No. 132014-21-2
Rilmakalim ( —— )
产品货号. M34129 CAS No. 132014-21-2
Rilmakalim (HOE 234) 是一种钾通道打开剂 (PCO)，可以激活心脏或其它组织中 ATP-敏感 K+ 通道。
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| 规格 | 价格/人民币 | 库存 | 数量 |
| 5MG | ￥2119 | 有现货 |
|
| 10MG | ￥3183 | 有现货 |
|
| 25MG | ￥5078 | 有现货 |
|
| 50MG | ￥7133 | 有现货 |
|
| 500MG | 获取报价 | 有现货 |
|
| 1G | 获取报价 | 有现货 |
|
生物学信息
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产品名称Rilmakalim
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注意事项本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
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产品简述Rilmakalim (HOE 234) 是一种钾通道打开剂 (PCO)，可以激活心脏或其它组织中 ATP-敏感 K+ 通道。
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产品描述Rilmakalim (HOE 234) is a potassium channel opener(PCO) that activates ATP-sensitive K+ channels in theheart or other tissues.
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体外实验——
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体内实验——
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同义词——
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通路Membrane Transporter/Ion Channel
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靶点Sodium Channel
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受体Sodium Channel
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研究领域——
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适应症——
化学信息
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CAS Number132014-21-2
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分子量401.48
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分子式C21H23NO5S
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纯度>98% (HPLC)
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溶解度——
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SMILESO[C@H]1[C@@H](C=2C(=CC=C(S(=O)(=O)C3=CC=CC=C3)C2)OC1(C)C)N4C(=O)CCC4
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化学全称——
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1. Kocic, Ivanet al. Hypotonic stress increases efficacy of rilmakalim, but not pinacidil, toactivate ATP-sensitive K(+) current in guinea pig ventricular myocytes. Journalof pharmacological sciences vol. 95,2 (2004): 189-95.?
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