Lesopitron
CAS No. 132449-46-8
Lesopitron ( —— )
产品货号. M34092 CAS No. 132449-46-8
Lesopitron is an anxiolytic with pre- and postsynaptic 5-HT1A agonist activity and is more effective than 5-HT1A agonists in rat social interaction and marmoset anxiety models. lesopitron counteracts benzodiazepine withdrawal-induced anxiety in rodents with low acute toxicity and does not potentiate the effects of alcohol or barbiturates.
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| 规格 | 价格/人民币 | 库存 | 数量 |
| 5MG | ¥2366 | 有现货 |
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| 10MG | ¥3534 | 有现货 |
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| 25MG | ¥5571 | 有现货 |
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| 50MG | ¥7710 | 有现货 |
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| 100MG | ¥9810 | 有现货 |
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| 500MG | ¥20070 | 有现货 |
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| 1G | 获取报价 | 有现货 |
|
| 1 mL x 10 mM in DMSO | ¥2242 | 有现货 |
|
生物学信息
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产品名称Lesopitron
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注意事项本公司产品仅用于科研实验,不得用于人体或动物的临床与诊断
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产品简述Lesopitron is an anxiolytic with pre- and postsynaptic 5-HT1A agonist activity and is more effective than 5-HT1A agonists in rat social interaction and marmoset anxiety models. lesopitron counteracts benzodiazepine withdrawal-induced anxiety in rodents with low acute toxicity and does not potentiate the effects of alcohol or barbiturates.
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产品描述Lesopitron is an anxiolytic with pre- and postsynaptic 5-HT1A agonist activity and is more effective than 5-HT1A agonists in rat social interaction and marmoset anxiety models. lesopitron counteracts benzodiazepine withdrawal-induced anxiety in rodents with low acute toxicity and does not potentiate the effects of alcohol or barbiturates.
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体外实验——
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体内实验——
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同义词——
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通路GPCR/G Protein
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靶点5-HT Receptor
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受体5-HT Receptor
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研究领域——
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适应症——
化学信息
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CAS Number132449-46-8
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分子量320.82
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分子式C15H21ClN6
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纯度>98% (HPLC)
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溶解度——
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SMILESC(CCCN1C=C(Cl)C=N1)N2CCN(CC2)C=3N=CC=CN3
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化学全称——
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
产品手册
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