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ICI 199,441 hydrochloride
CAS No. 115199-84-3
ICI 199,441 hydrochloride ( —— )
产品货号. M33868 CAS No. 115199-84-3
ICI 199441 是一种有效的选择性 κ-opioid 受体激动剂。ICI 199441 能提高心脏缺血/再灌注抵抗力。
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| 规格 | 价格/人民币 | 库存 | 数量 |
| 2MG | ￥261 | 有现货 |
|
| 5MG | ￥449 | 有现货 |
|
| 10MG | ￥701 | 有现货 |
|
| 25MG | ￥1386 | 有现货 |
|
| 50MG | ￥2223 | 有现货 |
|
| 100MG | ￥2871 | 有现货 |
|
| 200MG | ￥4032 | 有现货 |
|
| 500MG | 获取报价 | 有现货 |
|
| 1G | 获取报价 | 有现货 |
|
| 1 mL x 10 mM in DMSO | ￥528 | 有现货 |
|
生物学信息
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产品名称ICI 199,441 hydrochloride
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注意事项本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
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产品简述ICI 199441 是一种有效的选择性 κ-opioid 受体激动剂。ICI 199441 能提高心脏缺血/再灌注抵抗力。
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产品描述ICI 199441 is a potent and selective κ-opioid receptor agonist. ICI 199441 can improve heart resistance to ischemia/reperfusion.
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体外实验——
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体内实验ICI 199441 (Wistar rats, 0.1 mg/kg, IV, once) administered 15 min before ischemia produces a potent antiarrhythmic effect.
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同义词——
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通路Endocrinology/Hormones
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靶点Opioid Receptor
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受体Opioid Receptor
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研究领域——
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适应症——
化学信息
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CAS Number115199-84-3
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分子量427.8
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分子式C21H25Cl3N2O
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纯度>98% (HPLC)
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溶解度In Vitro:?DMSO 中的溶解度 : 250 mg/mL (584.39 mM; 超声助溶 )
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SMILESCl.CN([C@H](CN1CCCC1)c1ccccc1)C(=O)Cc1ccc(Cl)c(Cl)c1
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化学全称——
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1. Tsibulnikov SY, et al. Prospects of Using of κ-Opioid Receptor Agonists U-50,488 and ICI 199,441 for Improving Heart Resistance to Ischemia/Reperfusion. Bull Exp Biol Med. 2015;159(6):718-721.?
产品手册
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