SI-2 is an inhibitor (SMI) of steroid receptor coactivator-3 (SRC-3 or AIB1). SI-2 can selectively reduce the transcriptional activities and the protein concentrations of SRC-3 in cells, and selectively induce breast cancer cell death with IC50 values in the low nanomolar range (3-20 nM), but not affect normal cell viability.

Sisunatovir HCl 是一种口服的 RSV-F 蛋白抑制剂，在体外对一组 RSV-A 和 RSV-B 病毒临床分离株表现出强大的功效。

DAGLβ-IN-1 是一种通用中间体，用于设计 DAGL 定制的基于活性的探针，并且是二酰基甘油脂肪酶-β (DAGLβ) 的抑制剂。