Khellactone shows antitumor activity,it can suppress the growth of NCI-H460 tumor cells. (+)-4'-cis-Khellactone and (+)-3'-cis-khellactone have antiplasmodial activities, they show notable inhibitory activity against -sensitive strains of with IC(50) values from 1.5 and 2.4 microM.

Secretin (28-54), human, which acts on human secretin receptors, is a 27-amino acid residue C-terminally amidated peptide, .

TBOPP 是一种选择性 DOCK1 抑制剂 (IC50 : 8.4 μM)，对更广泛的肿瘤类型具有抗肿瘤活性。