Potent Nav1.7 blocker (IC50 = 2.5 nM). Also inhibits Nav1.1, Nav1.2, Nav1.3 and Nav1.6 in the nanomolar range. Exhibits no effects on Cav channels or nAChR at 5 μM. Demonstrates analgesic activity in vivo; antagonizes effects of scorpion-venom toxin OD1 at Nav1.7.

Limocitrin 3-β-D-glucose is a flavonoid glycoside.

PJ34 HCl 是 PJ34 的盐酸盐，PJ34 是一种 PARP 抑制剂，EC50 为 20 nM，与 PARP1/2 具有同等效力。