Oxyresveratrol 4,3',5'- tri-glucoside

Potent endogenous ligand of the kisspeptin receptor (KISS1, GPR54). Binds with high affinity to rat and human KISS1 receptors with Ki values of 1.80 and 1.45 nM respectively. Inhibits chemotaxis, invasion and metastasis of human melanomas and breast carcinomas. Stimulates gonadotropin secretion following i.c.v. administration.

1,1'-(4-氯丁亚基)双(4-氟苯)是Zerumbone的衍生物，对HeLa癌细胞具有潜在的抗肿瘤作用。