021-51111890
购物车（）
sales@molnova.cn
U 89843A
CAS No. 157013-32-6
U 89843A ( —— )
产品货号. M27731 CAS No. 157013-32-6
U 89843A 是 γ-氨基丁酸 (GABA)A 受体的正变构调节剂。
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| 规格 | 价格/人民币 | 库存 | 数量 |
| 5MG | ￥1691 | 有现货 |
|
| 10MG | ￥2518 | 有现货 |
|
| 25MG | ￥5506 | 有现货 |
|
| 50MG | ￥7700 | 有现货 |
|
| 100MG | ￥9450 | 有现货 |
|
| 500MG | 获取报价 | 有现货 |
|
| 1G | 获取报价 | 有现货 |
|
生物学信息
-
产品名称U 89843A
-
注意事项本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
-
产品简述U 89843A 是 γ-氨基丁酸 (GABA)A 受体的正变构调节剂。
-
产品描述U 89843A is a positive allosteric modulator of gamma-aminobutyric acid (GABA)A receptors.(In Vitro):In the alpha 1 beta 2 gamma 2 subtype of GABAA receptors expressed in human embryonic kidney cells, U 89843A dose-dependently enhanced 5 microM GABA-induced Cl- currents with a maximal enhancement of 362 +/- 91%, a half-maximal concentration of 2 +/- 0.4 microM and a slope factor of 1.1 +/- 0.4. U 89843A also inhibited [35S]t-butylbicyclophosphorothionate binding in rat cerebrocortical membranes with a similar half-maximal inhibitory concentration.
-
体外实验——
-
体内实验——
-
同义词——
-
通路Others
-
靶点Other Targets
-
受体acetylcholinesterase
-
研究领域——
-
适应症——
化学信息
-
CAS Number157013-32-6
-
分子量321.85
-
分子式C16H24ClN5
-
纯度>98% (HPLC)
-
溶解度——
-
SMILESCl.Cc1cc2c(nc(nc2n1C)N1CCCC1)N1CCCC1
-
化学全称——
运输与储存
-
储存条件(-20℃)
-
运输条件With Ice Pack
-
稳定性≥ 2 years
参考文献
1.Dafforn A, et al. Acetylcholinesterase inhibition by the ketone transition state analog phenoxyacetone and 1-halo-3-phenoxy-2-propanones. Biochem Biophys Res Commun. 1982 Jan 29;104(2):597-602.
产品手册
关联产品
-
Epinecidin-1
Epinecidin-1 (Piscidin-1 (22-42)) is a highly potent, multi-functional Antimicrobial Peptide (AMP) produced by Orange-spotted grouper (Epinephelus coioides). Epinecidin-1 has many functional usages including antibacterial, antifungal, antiviral, antiprotozoal, anticancer, immunomodulatory, and wound healing properties.
-
Ophiopogonone?C
Ophiopogonone C (compound 3) 是一种异黄酮类化合物，可从麦冬块茎的乙醇提取物中分离得到。
-
[Val4]-Angiotensin I...
[Val4] Angiotensin III 是一种血管紧张素 III 肽。[Val4] Angiotensin III 是一种有效的 Gαq 和 βarr2 反应的全激动剂，其 pEC50 值分别为 8.31 和 8.44。
