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Pranidipine
CAS No. 99522-79-9
Pranidipine ( OPC-13340 )
产品货号. M26794 CAS No. 99522-79-9
普拉地平是一种新型长效 1,4-二氢吡啶钙通道阻滞剂。
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| 规格 | 价格/人民币 | 库存 | 数量 |
| 5MG | ￥629 | 有现货 |
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| 10MG | ￥1007 | 有现货 |
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| 25MG | ￥1972 | 有现货 |
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| 50MG | ￥3143 | 有现货 |
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| 500MG | 获取报价 | 有现货 |
|
| 1G | 获取报价 | 有现货 |
|
| 1 mL x 10 mM in DMSO | ￥692 | 有现货 |
|
生物学信息
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产品名称Pranidipine
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注意事项本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
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产品简述普拉地平是一种新型长效 1,4-二氢吡啶钙通道阻滞剂。
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产品描述Pranidipine is a novel, long-acting 1,4-dihydropyridine calcium channel blocker. It prolongs acetylcholine-induced relaxation in presence of endothelium as well as nitroglycerin-induced relaxation in absence of endothelium. It also has antihypertensive activity.(In Vivo):Pranidipine enhances cyclic GMP-dependent nitric oxide-induced relaxation of rat aorta.
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体外实验——
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体内实验——
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同义词OPC-13340
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通路GPCR/G Protein
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靶点Calcium Channel
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受体Autophagy| mTORC1
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研究领域——
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适应症——
化学信息
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CAS Number99522-79-9
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分子量448.475
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分子式C25H24N2O6
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纯度>98% (HPLC)
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溶解度In Vitro:?DMSO : 270 mg/mL (602.05 mM)
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SMILESCOC(=O)C1=C(C)NC(C)=C(C1c1cccc(c1)[N+]([O-])=O)C(=O)OC\C=C\c1ccccc1
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化学全称——
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1.Laraia L, et al. The cholesterol transfer protein GRAMD1A regulates autophagosome biogenesis. Nat Chem Biol. 2019 Jul;15(7):710-720.
产品手册
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