Antihistamine-1 ( —— )

产品货号. M26056 CAS No. 1186430-60-3

COA

Datasheet

HNMR

HPLC

MSDS

Handing Instructions

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产品名称

Antihistamine-1
注意事项

本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
产品简述

Antihistamine-1 是一种 H1-抗组胺药（Ki：6.9 nM），具有可接受的血脑屏障渗透性，也是 CYP2D6 和 hERG 通道的抑制剂（IC50：5.4 和 0.8 μM）。
产品描述

Antihistamine-1 is an H1-antihistamine (Ki: 6.9 nM) with acceptable blood-brain barrier penetration and also an inhibitor of CYP2D6 and hERG channel (IC50s: 5.4 and 0.8 μM).(In Vitro):Antihistamine-1 is a H1-antihistamine (Ki=6.9 nM) with acceptable blood-brain barrier penetration and also an inhibitor of CYP2D6 and hERG channel with IC50s of 5.4 and 0.8 μM, respectively.
体外实验

Antihistamine-1 (Compound 2) is a H1-antihistamine (Ki=6.9 nM) with acceptable blood-brain barrier penetration and also an inhibitor of CYP2D6 and hERG channel with IC50s of 5.4 and 0.8 μM, respectively.
体内实验

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同义词

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通路

Metabolic Enzyme/Protease
靶点

P450
受体

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研究领域

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适应症

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计算器

产品手册

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