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ONC212
CAS No. 1807861-48-8
ONC212 ( —— )
产品货号. M20724 CAS No. 1807861-48-8
ONC212 是一种氟化 ONC201 类似物，是 GPR132 的选择性激动剂。
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| 规格 | 价格/人民币 | 库存 | 数量 |
| 5MG | ￥847 | 有现货 |
|
| 10MG | ￥1416 | 有现货 |
|
| 25MG | ￥2353 | 有现货 |
|
| 50MG | ￥3562 | 有现货 |
|
| 100MG | ￥4941 | 有现货 |
|
| 200MG | ￥6903 | 有现货 |
|
| 500MG | 获取报价 | 有现货 |
|
| 1G | 获取报价 | 有现货 |
|
| 1 mL x 10 mM in DMSO | ￥839 | 有现货 |
|
生物学信息
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产品名称ONC212
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注意事项本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
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产品简述ONC212 是一种氟化 ONC201 类似物，是 GPR132 的选择性激动剂。
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产品描述ONC212 a fluorinated-ONC201 analogue is a selective agonist of GPR132.
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体外实验——
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体内实验——
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同义词——
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通路GPCR/G Protein
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靶点GHSR
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受体GPR132
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研究领域——
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适应症——
化学信息
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CAS Number1807861-48-8
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分子量440.46
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分子式C24H23F3N4O
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纯度>98% (HPLC)
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溶解度DMSO:50 mg/mL (113.52 mM)
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SMILESFC(F)(F)c1ccc(CN2C3=NCCN3C3=C(CN(Cc4ccccc4)CC3)C2=O)cc1
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化学全称246789-Hexahydro-7-(phenylmethyl)-4-[[4-(trifluoromethyl)phenyl]methyl]imidazo[12-a]pyrido[34-e]pyrimidin-5(1H)-one
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1.Nii T Prabhu VV Ruvolo Vet al.Imipridone ONC212 activates orphan G protein-coupled receptor GPR132 and integrated stress response in acute myeloid leukemia[J].Leukemia. 2019 Dec;33(12):2805-2816.
产品手册
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