021-51111890
购物车（）
sales@molnova.cn
Bepridil hydrochloride
CAS No. 68099-86-5
Bepridil hydrochloride ( CERM 1978 )
产品货号. M20140 CAS No. 68099-86-5
Bepridil 是一种钙通道阻滞剂，还抑制 Na+/Ca2+ 交换 (NCX)、钠通道和心脏肌膜 KATP 通道。
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| 规格 | 价格/人民币 | 库存 | 数量 |
| 2MG | ￥238 | 有现货 |
|
| 5MG | ￥396 | 有现货 |
|
| 10MG | ￥554 | 有现货 |
|
| 25MG | ￥918 | 有现货 |
|
| 50MG | ￥1376 | 有现货 |
|
| 100MG | ￥1998 | 有现货 |
|
| 200MG | ￥2997 | 有现货 |
|
| 500MG | 获取报价 | 有现货 |
|
| 1G | 获取报价 | 有现货 |
|
| 1 mL x 10 mM in DMSO | ￥433 | 有现货 |
|
生物学信息
-
产品名称Bepridil hydrochloride
-
注意事项本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
-
产品简述Bepridil 是一种钙通道阻滞剂，还抑制 Na+/Ca2+ 交换 (NCX)、钠通道和心脏肌膜 KATP 通道。
-
产品描述Bepridil is a calcium channel blocker and also inhibits Na+/Ca2+ exchange (NCX) sodium channels and cardiac sarcolemmal KATP channels.(In Vitro):Bepridil hydrochloride is a calcium channel blocker, with antianginal activity.(In Vivo):Bepridil hydrochloride (21 mg/kg) reduces heart rate and mean arterial pressure, decreases the mean coronary vascular resistance and increases stroke volume in rats.
-
体外实验Bepridil hydrochloride is a calcium channel blocker, with antianginal activity.
-
体内实验Bepridil hydrochloride (21 mg/kg) reduces heart rate and mean arterial pressure, decreases the mean coronary vascular resistance and increases stroke volume in rats.
-
同义词CERM 1978
-
通路GPCR/G Protein
-
靶点Calcium Channel
-
受体Calcium Channel
-
研究领域Cardiovascular Disease
-
适应症Angina pectoris; Tachycardia
化学信息
-
CAS Number68099-86-5
-
分子量403
-
分子式C24H35ClN2O
-
纯度>98% (HPLC)
-
溶解度DMSO: 130 mg/mL (322.58 mM)
-
SMILESCl.CC(C)COCC(CN(Cc1ccccc1)c1ccccc1)N1CCCC1
-
化学全称——
运输与储存
-
储存条件(-20℃)
-
运输条件With Ice Pack
-
稳定性≥ 2 years
参考文献
1.Flaim SF et al. Effects of bepridil hydrochloride on cardiocirculatory dynamics coronary vascular resistance and cardiac output distribution in normal conscious rats. J Cardiovasc Pharmacol. 1988 Mar;11(3):363-72.
产品手册
关联产品
-
Strophanthidin
旋花草苷可诱导体内钙超载。
-
Cav 2.2 blocker 1
Cav 2.2 blocker 1 是一种 N 型钙通道 (Cav 2.2; IC50: 1 nM) 阻断剂，用于治疗疼痛。
-
Verapamil hydrochlor...
Verapamil Hcl 是一种苯烷基胺类 L 型钙通道阻滞剂。
