Bilastine

本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断

比拉斯汀是一种新型新一代抗组胺药，对H1组胺受体具有高度选择性，起效快，作用持续时间长。

Bilastine (trade name Bilaxten) is a second generation antihistamine drug for the treatment of allergic rhinoconjunctivitis and urticaria (hives). It exerts its effect as a selective histamine H1 receptor antagonist, and has a potency similar to cetirizine and is superior to fexofenadine. It was developed in Spain by FAES Farma. Bilastine is approved in the European Union for the symptomatic treatment of allergic rhinoconjunctivitis and urticaria, but it is not approved by the U.S. Food and Drug Administration for any use in the United States. Bilastine has been effective in the treatment of ocular symptoms and diseases of allergies, including rhinoconjuctivitis. Additionally, bilastine has been shown to improve quality of life, and all nasal and ocular symptoms related to allergic rhinitis.

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Bilastine trade name Bilaxten

Endocrinology/Hormones

5-HT Receptor

H1 receptor

Inflammation/Immunology

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202189-78-4

463.62

C28H37N3O3

>98% (HPLC)

DMSO : ≥ 49.3 mg/mL; 106.34 mM

CCOCCn1c(nc2ccccc12)C1CCN(CCc2ccc(cc2)C(C)(C)C(O)=O)CC1

2-(4-(2-(4-(1-(2-ethoxyethyl)-1H-benzo[d]imidazol-2-yl)piperidin-1-yl)ethyl)phenyl)-2-methylpropanoic acid

(-20℃)

With Ice Pack

≥ 2 years