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Cisatracurium besylate

CAS No. 96946-42-8

Cisatracurium besylate ( —— )

产品货号. M16875 CAS No. 96946-42-8

Cisatracurium Besylate 是一种用于静脉注射的非去极化骨骼肌松弛剂。

纯度: >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
规格 价格/人民币 库存 数量
5MG ¥269 有现货
10MG ¥375 有现货
25MG ¥617 有现货
50MG ¥1014 有现货
100MG ¥1458 有现货
200MG ¥2178 有现货
500MG ¥3537 有现货
1G 获取报价 有现货
1 mL x 10 mM in DMSO ¥499 有现货

生物学信息

  • 产品名称
    Cisatracurium besylate
  • 注意事项
    本公司产品仅用于科研实验,不得用于人体或动物的临床与诊断
  • 产品简述
    Cisatracurium Besylate 是一种用于静脉注射的非去极化骨骼肌松弛剂。
  • 产品描述
    Cisatracurium Besylate is a nondepolarizing skeletal muscle relaxant for intravenous administration. Cisatracurium Besylate acts on cholinergic receptors, blocking neuromuscular transmission. This action is antagonized by acetylcholinesterase inhibitors such as neostigmine. The neuromuscular block produced by cisatracurium besylate is readily antagonized by anticholinesterase agents once recovery has started. As with other nondepolarizing neuromuscular blocking agents, the more profound the neuromuscular block at the time of reversal, the longer the time required for recovery of neuromuscular function. Compared to other neuromuscular blocking agents, it is intermediate in its onset and duration of action. (In Vitro):Cisatracurium Besylate (51W89) is a neuromuscular-blocking drug or skeletal muscle relaxant in the category of non-depolarizing neuromuscular-blocking drugs, used adjunctively in anesthesia to facilitate endotracheal intubation and to provide skeletal muscle relaxation during surgery or mechanical ventilation. It is a bisbenzyltetrahydroisoquinolinium agent with an intermediate duration of action. Cisatracurium Besylate (51W89) is one of the ten isomers of the parent molecule, atracurium. Moreover, cisatracurium represents approximately 15% of the atracurium mixture.
  • 体外实验
    Cisatracurium Besylate (51W89) is a neuromuscular-blocking drug or skeletal muscle relaxant in the category of non-depolarizing neuromuscular-blocking drugs, used adjunctively in anesthesia to facilitate endotracheal intubation and to provide skeletal muscle relaxation during surgery or mechanical ventilation. It is a bisbenzyltetrahydroisoquinolinium agent with an intermediate duration of action. Cisatracurium Besylate (51W89) is one of the ten isomers of the parent molecule, atracurium. Moreover, cisatracurium represents approximately 15% of the atracurium mixture.
  • 体内实验
    ——
  • 同义词
    ——
  • 通路
    Endocrinology/Hormones
  • 靶点
    AChR
  • 受体
    AChR| Adrenergic Receptor
  • 研究领域
    Neurological Disease
  • 适应症
    ——

化学信息

  • CAS Number
    96946-42-8
  • 分子量
    1243.48
  • 分子式
    C53H72N2O12·2C6H5O3S
  • 纯度
    >98% (HPLC)
  • 溶解度
    Ethanol: 249 mg/mL (200.24 mM); Water: 47 mg/mL (37.79 mM); DMSO: 249 mg/mL (200.24 mM)
  • SMILES
    C[N@@+]1(CCC2=CC(=C(C=C2[C@H]1CC3=CC(=C(C=C3)OC)OC)OC)OC)CCC(=O)OCCCCCOC(=O)CC[N@+]4(CCC5=CC(=C(C=C5[C@H]4CC6=CC(=C(C=C6)OC)OC)OC)OC)C.C1=CC=C(C=C1)S(=O)(=O)[O-].C1=CC=C(C=C1)S(=O)(=O)[O-]
  • 化学全称
    ——

运输与储存

  • 储存条件
    (-20℃)
  • 运输条件
    With Ice Pack
  • 稳定性
    ≥ 2 years

参考文献

1.Dieye E, et al. Ann Intensive Care. 2014 Feb 11;4(1):3.
产品手册
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