Moracin M, a phenolic component in the skin of Morus alba Linn., is a potent phosphodiesterase-4 (PDE4) inhibitor with IC50 values of 2.9, 4.5, >40, and >100 μM for PDE4D2, PDE4B2, PDE5A1, and PDE9A2, respectively. Moracin M has anti-inflammatory activity.

The a-helix of the amphipathic peptide antibiotic LAH4 (KKALLALALHHLAHLALHLALALKKA-NH2) strongly interacts with phospholipid membranes, demonstrating in vitro transfection efficiencies comparable to those of commercially available reagents.

yGsy2p-IN-1 是一种有效的酵母糖原合酶 2 (yGsy2p) 和人糖原合酶 1 (hGYS1) 抑制剂。 yGsy2p-IN-H23 一种吡唑抑制剂，用于治疗糖原贮积病 (GSD)。