Carvedilol phosphate
CAS No. 610309-89-2
Carvedilol phosphate ( —— )
产品货号. M15292 CAS No. 610309-89-2
卡维地洛是一种非选择性β受体阻滞剂,适用于治疗轻度至中度充血性心力衰竭(CHF)。
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| 规格 | 价格/人民币 | 库存 | 数量 |
| 25MG | ¥117 | 有现货 |
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| 50MG | ¥184 | 有现货 |
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| 100MG | ¥320 | 有现货 |
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| 500MG | ¥669 | 有现货 |
|
| 1G | 获取报价 | 有现货 |
|
生物学信息
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产品名称Carvedilol phosphate
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注意事项本公司产品仅用于科研实验,不得用于人体或动物的临床与诊断
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产品简述卡维地洛是一种非选择性β受体阻滞剂,适用于治疗轻度至中度充血性心力衰竭(CHF)。
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产品描述Carvedilol is a non-selective beta blocker indicated in the treatment of mild to moderate congestive heart failure (CHF). It blocks beta-1 and beta-2 adrenergic receptors as well as the alpha-1 adrenergic receptors.
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体外实验Superoxide generation by activated human neutrophils in vitro is inhibited by Carvedilol with an IC50 of 28 μM. Carvedilol is shown to scavenge oxygen free radicals in a cell-free system with an IC50 of 25 μM.
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体内实验——
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同义词——
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通路Endocrinology/Hormones
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靶点Adrenergic Receptor
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受体Adrenergic Receptor| Gap Junction Protein| E-selectin| NADPH dehydrogenase| Natriuretic peptides B| VCAM1| Potassium Channel| VEGFR
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研究领域Cardiovascular Disease
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适应症——
化学信息
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CAS Number610309-89-2
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分子量522.49
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分子式C24H26N2O4·H2O·H3O4P
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纯度>98% (HPLC)
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溶解度Water: 10 mM
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SMILESO.OP(O)(O)=O.COC1=CC=CC=C1OCCNCC(O)COC1=CC=CC2=C1C1=CC=CC=C1N2
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化学全称——
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1.Nichols AJ, et al. Fundam Clin Pharmacol. 1991;5(1):25-38.
产品手册
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