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Flopropione

CAS No. 2295-58-1

Flopropione ( —— )

产品货号. M13637 CAS No. 2295-58-1

Flopropione 是一种解痉剂或解痉剂,可作为 5-HT1A 受体拮抗剂。

纯度: >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
规格 价格/人民币 库存 数量
50MG ¥184 有现货
100MG ¥260 有现货
200MG ¥372 有现货
500MG ¥611 有现货
1G 获取报价 有现货
1 mL x 10 mM in DMSO ¥302 有现货

生物学信息

  • 产品名称
    Flopropione
  • 注意事项
    本公司产品仅用于科研实验,不得用于人体或动物的临床与诊断
  • 产品简述
    Flopropione 是一种解痉剂或解痉剂,可作为 5-HT1A 受体拮抗剂。
  • 产品描述
    Flopropione is a spasmolytic or antispasmodic agent, and acts as a 5-HT1A receptor antagonist(In Vivo):The effect of Flopropione as an antispasmodic agent on the rate of passing a calculus from the urinary tract has been compared retrospectively with patients in whom passage was spontaneous. Flopropine has been shown, with statistical significance, to be superior to the control in cumulative passage rate after initiation of administration. Flopropine has been shown to exert a spasmolytic effect not only on smooth muscle of the gastrointestinal tract but also on smooth muscle of the pancreatobiliary and urinary systems.
  • 体外实验
    ——
  • 体内实验
    The effect of Flopropione as an antispasmodic agent on the rate of passing a calculus from the urinary tract has been compared retrospectively with patients in whom passage was spontaneous. Flopropine has been shown, with statistical significance, to be superior to the control in cumulative passage rate after initiation of administration. Flopropine has been shown to exert a spasmolytic effect not only on smooth muscle of the gastrointestinal tract but also on smooth muscle of the pancreatobiliary and urinary systems.
  • 同义词
    ——
  • 通路
    Endocrinology/Hormones
  • 靶点
    5-HT Receptor
  • 受体
    5-HT1A
  • 研究领域
    Neurological Disease
  • 适应症
    ——

化学信息

  • CAS Number
    2295-58-1
  • 分子量
    182.18
  • 分子式
    C9H10O4
  • 纯度
    >98% (HPLC)
  • 溶解度
    Ethanol: 36 mg/mL (197.61 mM); DMSO: 36 mg/mL (197.61 mM)
  • SMILES
    CCC(=O)C1=C(O)C=C(O)C=C1O
  • 化学全称
    ——

运输与储存

  • 储存条件
    (-20℃)
  • 运输条件
    With Ice Pack
  • 稳定性
    ≥ 2 years

参考文献

1.Aso Y, et al. J Pharm Sci, 2000, 89(3), 408-416.
产品手册
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