Leptomerine ( —— )

产品货号. M29180 CAS No. 22048-97-1

COA

Datasheet

HNMR

HPLC

MSDS

Handing Instructions

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产品名称

Leptomerine
注意事项

本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
产品简述

Leptomerine 是一种来自 Esenbeckia leiocarpa Engl 茎的生物碱。（芸香科）。 Leptomerine 显示出抗胆碱酯酶活性，可用于阿尔茨海默病研究。
产品描述

Leptomerine is an alkaloid from stems of Esenbeckia leiocarpa Engl. (Rutaceae). Leptomerine shows as anticholinesterasic activity and can be used in Alzheimer Disease studies.(In Vitro):Bioactivity-guided fractionation of the ethanol stems extract afforded the isolation of six alkaloids: leiokinine A, Leptomerine, kokusaginine, skimmianine, maculine and flindersiamine. The alkaloid Leptomerine showed the highest activity (IC50 = 2.5 mM), similar to that of the reference compound galanthamine (IC50 = 1.7 mM).
体外实验

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体内实验

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同义词

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通路

Metabolic Enzyme/Protease
靶点

AChE
受体

AChE
研究领域

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适应症

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计算器

产品手册

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