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HA155
CAS No. 1312201-00-5
HA155 ( CS-963 )
产品货号. M26244 CAS No. 1312201-00-5
HA155 选择性且有效地抑制自分泌运动因子，IC50 为 5.7 nM。
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| 规格 | 价格/人民币 | 库存 | 数量 |
| 5MG | ￥3013 | 有现货 |
|
| 10MG | ￥4447 | 有现货 |
|
| 25MG | ￥7039 | 有现货 |
|
| 50MG | ￥9477 | 有现货 |
|
| 100MG | ￥12798 | 有现货 |
|
| 200MG | 获取报价 | 有现货 |
|
| 500MG | 获取报价 | 有现货 |
|
| 1G | 获取报价 | 有现货 |
|
生物学信息
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产品名称HA155
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注意事项本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
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产品简述HA155 选择性且有效地抑制自分泌运动因子，IC50 为 5.7 nM。
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产品描述HA155 selectively and potently inhibits autotaxin with an IC50 of 5.7 nM.(In Vitro):HA155 completely attenuates the thrombin-mediated increase in platelet-derived LPA dose-dependently .HA155 is an ATX inhibitor by binding to the ATX active site .
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体外实验HA-155 inhibits ATX by binding to the ATX active site.HA155 completely attenuates the thrombin-mediated increase in platelet-derived LPA in a dose-dependent manner.
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体内实验——
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同义词CS-963
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通路Angiogenesis
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靶点PDE
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受体Antibacterial
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研究领域——
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适应症——
化学信息
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CAS Number1312201-00-5
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分子量463.29
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分子式C24H19BFNO5S
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纯度>98% (HPLC)
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溶解度In Vitro:?DMSO : 10 mg/mL (21.58 mM)
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SMILESO=C1N(CC2=CC=C(F)C=C2)C(S/C1=C\C3=CC=C(OCC4=CC=C(B(O)O)C=C4)C=C3)=O.[(Z)]
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化学全称——
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1.Guo B, et al. Clinical Pharmacokinetics of Levornidazole in Elderly Subjects and Dosing Regimen Evaluation Using Pharmacokinetic/Pharmacodynamic Analysis. Clin Ther. 2017 Jul;39(7):1336-1346.
产品手册
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