Eslicarbazepine ( BIA 2-194 )

产品货号. M27993 CAS No. 104746-04-5

COA

Datasheet

HNMR

HPLC

MSDS

Handing Instructions

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产品名称

Eslicarbazepine
注意事项

本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
产品简述

艾斯利卡西平可用于成人部分性癫痫发作的辅助治疗。
产品描述

Eslicarbazepine can be used for adjunctive therapy for adults with partial-onset seizures.(In Vitro):Eslicarbazepine is an anti-epileptic drug, chemically related to carbamazepine but with a more favorable safety profile. Eslicarbazepine acetate is a prodrug for eslicarbazepine (S-licarbazepine), which is a dual Inhibitor of β-Secretase and voltage-gated sodium channel.
体外实验

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体内实验

Eslicarbazepine is an anti-epileptic drug, chemically related to carbamazepine but with a more favorable safety profile. Eslicarbazepine acetate is a prodrug for eslicarbazepine (S-licarbazepine), which is a dual a dual Inhibitor of β-Secretase and voltage-gated sodium channel.
同义词

BIA 2-194
通路

Membrane Transporter/Ion Channel
靶点

Sodium Channel
受体

Chitotriosidase (CHIT1)
研究领域

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适应症

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1.Mazur M, et al. Discovery of selective, orally bioavailable inhibitor of mouse chitotriosidase. Bioorg Med Chem Lett. 2018 Feb 1;28(3):310-314.

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