Antide

本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断

Antide (D-21074) 是一种有效的 LHRH 拮抗剂。Antide 也可用于前列腺癌的研究。

Antide (D-21074) is a potent LHRH antagonist. Antide also can be used for the research of prostatic cancer.

Antide（皮下注射；1、3、6、10 和 15 mg/kg；一次或连续 5 天）可引起成年雄性大鼠和食蟹猴的长期化学阉割。Animal Model:Cynomolgus monkey and rat Dosage:1, 3, 6, 10 and 15 mg/kg Administration:Subcutaneous, once or on 5 consecutive days Result:Had a dose-dependent inhibitory effect on serum concentration of LH (only rat) and testosterone and on the weights of the testes, prostates and seminal vesicles.Achieved long-lasting castration-like effects at concentrations between 6 (less than or equal to 8 weeks) and 15 mg/kg (greater than 8 weeks) in the rat. Induced a prolonged inhibitory effect only at 15 mg/kg and the duration was only 2-3 weeks in the cynomolgus monkey.

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Others

Other Targets

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112568-12-4

1591.29

C82H108ClN17O14

>98% (HPLC)

H2O : 10 mg/mL (6.28 mM; ultraphonic)

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(-20℃)

With Ice Pack

≥ 2 years